Receptor Information
General Information of This Receptor
| Receptor ID |
REC00064
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| Receptor Name |
Falcipain-1 (FP1)
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| Gene Name |
FP1
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| Gene ID | ||||||
| Synonym |
Cysteine proteinase falcipain-1 ; Trophozoite cysteine proteinase
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| Sequence |
MVAIKEMKEFAFARPSLVETLNKKKKFLKKKEKRTFVLSIYAFITFIIFCIGILYFTNKS
SAHNNNNNKNEHSLKKEEIELLRVLLEKYKKQKDGILNESSNEEDEEKYTLNSETYNNKN NVSNIKNDSIKSKKEEYINLERILLEKYKKFINENNEENRKELSNILHKLLEINKLILRE EKDDKKVYLINDNYDEKGALEIGMNEEMKYKKEDPINNIKYASKFFKFMKEHNKVYKNID EQMRKFEIFKINYISIKNHNKLNKNAMYKKKVNQFSDYSEEELKEYFKTLLHVPNHMIEK YSKPFENHLKDNILISEFYTNGKRNEKDIFSKVPEILDYREKGIVHEPKDQGLCGSCWAF ASVGNIESVFAKKNKNILSFSEQEVVDCSKDNFGCDGGHPFYSFLYVLQNELCLGDEYKY KAKDDMFCLNYRCKRKVSLSSIGAVKENQLILALNEVGPLSVNVGVNNDFVAYSEGVYNG TCSEELNHSVLLVGYGQVEKTKLNYNNKIQTYNTKENSNQPDDNIIYYWIIKNSWSKKWG ENGFMRLSRNKNGDNVFCGIGEEVFYPIL
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| 3D Structure | ||||||
| Family |
the peptidase C1 family
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| Function |
Cysteine protease. In the mosquito midgut, required for parasite development.
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| Uniprot Entry | ||||||
| KEGG ID | ||||||
Each Peptide-drug Conjuate AND It's Component Related to This Receptor
Full List of The PDC Related to This Receptor
LFX 8a
| PDC Info | PDC Name | Drug | Target | Linker |
|---|---|---|---|---|
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Dipeptide 23 - 4-Amino-7-chloroquinoline conjugate 10
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4-Amino-7-chloroquinoline
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Undisclosed
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Amide bond
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LFX 8b
| PDC Info | PDC Name | Drug | Target | Linker |
|---|---|---|---|---|
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Dipeptide 23 - 4-Amino-7-chloroquinoline conjugate 9
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4-Amino-7-chloroquinoline
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Undisclosed
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Amide bond
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LFX 8c
| PDC Info | PDC Name | Drug | Target | Linker |
|---|---|---|---|---|
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Dipeptide 23 - 4-Amino-7-chloroquinoline conjugate 8
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4-Amino-7-chloroquinoline
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Undisclosed
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Amide bond
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LFX 8d
| PDC Info | PDC Name | Drug | Target | Linker |
|---|---|---|---|---|
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Dipeptide 23 - 4-Amino-7-chloroquinoline conjugate 7
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4-Amino-7-chloroquinoline
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Undisclosed
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Amide bond
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LFX 8e
| PDC Info | PDC Name | Drug | Target | Linker |
|---|---|---|---|---|
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Dipeptide 23 - 4-Amino-7-chloroquinoline conjugate 12
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4-Amino-7-chloroquinoline
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Undisclosed
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Amide bond
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LFX 8f
| PDC Info | PDC Name | Drug | Target | Linker |
|---|---|---|---|---|
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Dipeptide 23 - 4-Amino-7-chloroquinoline conjugate 6
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4-Amino-7-chloroquinoline
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Undisclosed
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Amide bond
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LFX 8h
| PDC Info | PDC Name | Drug | Target | Linker |
|---|---|---|---|---|
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Dipeptide 23 - 4-Amino-7-chloroquinoline conjugate 5
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4-Amino-7-chloroquinoline
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Undisclosed
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Amide bond
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LFX 8i
| PDC Info | PDC Name | Drug | Target | Linker |
|---|---|---|---|---|
|
Dipeptide 23 - 4-Amino-7-chloroquinoline conjugate 4
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4-Amino-7-chloroquinoline
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Undisclosed
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Amide bond
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LFX 8k
| PDC Info | PDC Name | Drug | Target | Linker |
|---|---|---|---|---|
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Dipeptide 23 - 4-Amino-7-chloroquinoline conjugate 1
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4-Amino-7-chloroquinoline
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Undisclosed
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Amide bond
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